KIT

ENSG00000157404 - H. sapiens

Pathways

Go term Description
GO:0002020 protease binding
GO:0004713 protein tyrosine kinase activity
GO:0004714 transmembrane receptor protein tyrosine kinase activity
GO:0004716 signal transducer, downstream of receptor, with protein tyrosine kinase activity
GO:0005020 stem cell factor receptor activity
GO:0005088 Ras guanyl-nucleotide exchange factor activity
GO:0005515 protein binding
GO:0005524 ATP binding
GO:0019955 cytokine binding
GO:0042803 protein homodimerization activity
GO:0046872 metal ion binding
GO:0046934 phosphatidylinositol-4,5-bisphosphate 3-kinase activity

Drugs

Drug name Description
CABOZANTINIB
DASATINIB Tyrosine-protein kinase ABL inhibitor
IMATINIB Tyrosine-protein kinase ABL inhibitor
LENVATINIB
PAZOPANIB Tyrosine-protein kinase LCK inhibitor
PONATINIB Tyrosine-protein kinase ABL inhibitor
REGORAFENIB Tyrosine-protein kinase ABL inhibitor
SORAFENIB Serine/threonine-protein kinase RAF inhibitor
SUNITINIB Macrophage colony stimulating factor receptor inhibitor

Diseases

Disease Name
GIST
AML
TGCT
mastocytosis
mucosal melanoma
epithelioma

Orthologs

Gene Organism
Pvr D. melanogaster

Related Interactions

Gene ID A Gene Name A Gene ID B Gene Symbol B Organism Source Score?
ENSG00000149269 PAK1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.931961 View
ENSG00000092421 SEMA6A ENSG00000157404 KIT H. sapiens SDL Slorth 0.931824 View
ENSG00000111262 KCNA1 ENSG00000157404 KIT H. sapiens SDL Slorth 0.931688 View
ENSG00000089159 PXN ENSG00000157404 KIT H. sapiens SSL Slorth 0.931512 View
ENSG00000067141 NEO1 ENSG00000157404 KIT H. sapiens SDL Slorth 0.931303 View
ENSG00000126261 UBA2 ENSG00000157404 KIT H. sapiens SSL Slorth 0.931246 View
ENSG00000088367 EPB41L1 ENSG00000157404 KIT H. sapiens SDL Slorth 0.930835 View
ENSG00000066468 FGFR2 ENSG00000157404 KIT H. sapiens SSL Slorth 0.930642 View
ENSG00000133124 IRS4 ENSG00000157404 KIT H. sapiens SDL Slorth 0.930492 View
ENSG00000117676 RPS6KA1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.93042 View
ENSG00000117400 MPL ENSG00000157404 KIT H. sapiens SDL Slorth 0.930336 View
ENSG00000135312 HTR1B ENSG00000157404 KIT H. sapiens SDL Slorth 0.930336 View
ENSG00000141503 MINK1 ENSG00000157404 KIT H. sapiens SDL Slorth 0.9303 View
ENSG00000139998 RAB15 ENSG00000157404 KIT H. sapiens SDL Slorth 0.930244 View
ENSG00000115592 PRKAG3 ENSG00000157404 KIT H. sapiens SDL Slorth 0.930244 View
ENSG00000106327 TFR2 ENSG00000157404 KIT H. sapiens SDL Slorth 0.930244 View
ENSG00000010810 FYN ENSG00000157404 KIT H. sapiens SDL Slorth 0.929851 View
ENSG00000072736 NFATC3 ENSG00000157404 KIT H. sapiens SDL Slorth 0.929846 View
ENSG00000117399 CDC20 ENSG00000157404 KIT H. sapiens SSL Slorth 0.929719 View
ENSG00000155465 SLC7A7 ENSG00000157404 KIT H. sapiens SDL Slorth 0.929631 View
ENSG00000157106 SMG1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.929608 View
ENSG00000143252 SDHC ENSG00000157404 KIT H. sapiens SDL Slorth 0.92921 View
ENSG00000061918 GUCY1B3 ENSG00000157404 KIT H. sapiens SDL Slorth 0.928957 View
ENSG00000120438 TCP1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.928582 View
ENSG00000157404 KIT ENSG00000254087 LYN H. sapiens SSL Slorth 0.928373 View
ENSG00000157404 KIT ENSG00000213341 CHUK H. sapiens SSL Slorth 0.928359 View
ENSG00000073111 MCM2 ENSG00000157404 KIT H. sapiens SSL Slorth 0.927876 View
ENSG00000135018 UBQLN1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.927681 View
ENSG00000152822 GRM1 ENSG00000157404 KIT H. sapiens SDL Slorth 0.927654 View
ENSG00000006451 RALA ENSG00000157404 KIT H. sapiens SSL Slorth 0.927214 View
ENSG00000146094 DOK3 ENSG00000157404 KIT H. sapiens SDL Slorth 0.927052 View
ENSG00000066455 GOLGA5 ENSG00000157404 KIT H. sapiens SDL Slorth 0.926925 View
ENSG00000154229 PRKCA ENSG00000157404 KIT H. sapiens SSL Slorth 0.926501 View
ENSG00000157404 KIT ENSG00000177885 GRB2 H. sapiens SDL Slorth 0.926465 View
ENSG00000141480 ARRB2 ENSG00000157404 KIT H. sapiens SSL Slorth 0.926175 View
ENSG00000039068 CDH1 ENSG00000157404 KIT H. sapiens SDL Slorth 0.925602 View
ENSG00000051382 PIK3CB ENSG00000157404 KIT H. sapiens SSL Slorth 0.925464 View
ENSG00000100982 PCIF1 ENSG00000157404 KIT H. sapiens SDL Slorth 0.92533 View
ENSG00000157404 KIT ENSG00000165671 NSD1 H. sapiens SDL Slorth 0.925118 View
ENSG00000041353 RAB27B ENSG00000157404 KIT H. sapiens SDL Slorth 0.924748 View