KIT

ENSG00000157404 - H. sapiens

Pathways

Go term Description
GO:0002020 protease binding
GO:0004713 protein tyrosine kinase activity
GO:0004714 transmembrane receptor protein tyrosine kinase activity
GO:0004716 signal transducer, downstream of receptor, with protein tyrosine kinase activity
GO:0005020 stem cell factor receptor activity
GO:0005088 Ras guanyl-nucleotide exchange factor activity
GO:0005515 protein binding
GO:0005524 ATP binding
GO:0019955 cytokine binding
GO:0042803 protein homodimerization activity
GO:0046872 metal ion binding
GO:0046934 phosphatidylinositol-4,5-bisphosphate 3-kinase activity

Drugs

Drug name Description
CABOZANTINIB
DASATINIB Tyrosine-protein kinase ABL inhibitor
IMATINIB Tyrosine-protein kinase ABL inhibitor
LENVATINIB
PAZOPANIB Tyrosine-protein kinase LCK inhibitor
PONATINIB Tyrosine-protein kinase ABL inhibitor
REGORAFENIB Tyrosine-protein kinase ABL inhibitor
SORAFENIB Serine/threonine-protein kinase RAF inhibitor
SUNITINIB Macrophage colony stimulating factor receptor inhibitor

Diseases

Disease Name
GIST
AML
TGCT
mastocytosis
mucosal melanoma
epithelioma

Orthologs

Gene Organism
Pvr D. melanogaster

Related Interactions

Gene ID A Gene Name A Gene ID B Gene Symbol B Organism Source Score?
ENSG00000100030 MAPK1 ENSG00000157404 KIT H. sapiens SDL Slorth 0.941726 View
ENSG00000157404 KIT ENSG00000185022 MAFF H. sapiens SDL Slorth 0.941715 View
ENSG00000137486 ARRB1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.941384 View
ENSG00000115221 ITGB6 ENSG00000157404 KIT H. sapiens SDL Slorth 0.941366 View
ENSG00000026103 FAS ENSG00000157404 KIT H. sapiens SSL Slorth 0.940205 View
ENSG00000110330 BIRC2 ENSG00000157404 KIT H. sapiens SSL Slorth 0.9401 View
ENSG00000157404 KIT ENSG00000169083 AR H. sapiens SDL Slorth 0.939922 View
ENSG00000125810 CD93 ENSG00000157404 KIT H. sapiens SDL Slorth 0.939522 View
ENSG00000128908 INO80 ENSG00000157404 KIT H. sapiens SSL Slorth 0.939281 View
ENSG00000116030 SUMO1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.938098 View
ENSG00000010810 FYN ENSG00000157404 KIT H. sapiens SSL Slorth 0.937961 View
ENSG00000105974 CAV1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.937532 View
ENSG00000067606 PRKCZ ENSG00000157404 KIT H. sapiens SSL Slorth 0.936879 View
ENSG00000157404 KIT ENSG00000186868 MAPT H. sapiens SSL Slorth 0.936737 View
ENSG00000021574 SPAST ENSG00000157404 KIT H. sapiens SDL Slorth 0.936553 View
ENSG00000061273 HDAC7 ENSG00000157404 KIT H. sapiens SSL Slorth 0.936301 View
ENSG00000079156 OSBPL6 ENSG00000157404 KIT H. sapiens SDL Slorth 0.936277 View
ENSG00000148248 SURF4 ENSG00000157404 KIT H. sapiens SDL Slorth 0.936021 View
ENSG00000157404 KIT ENSG00000183791 TCEB3C H. sapiens SDL Slorth 0.935896 View
ENSG00000141968 VAV1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.935212 View
ENSG00000099785 MARCH2 ENSG00000157404 KIT H. sapiens SDL Slorth 0.935165 View
ENSG00000157404 KIT ENSG00000182511 FES H. sapiens SDL Slorth 0.934932 View
ENSG00000136238 RAC1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.934748 View
ENSG00000129245 FXR2 ENSG00000157404 KIT H. sapiens SDL Slorth 0.934575 View
ENSG00000097007 ABL1 ENSG00000157404 KIT H. sapiens SDL Slorth 0.934526 View
ENSG00000105810 CDK6 ENSG00000157404 KIT H. sapiens SSL Slorth 0.934223 View
ENSG00000135624 CCT7 ENSG00000157404 KIT H. sapiens SSL Slorth 0.93355 View
ENSG00000085511 MAP3K4 ENSG00000157404 KIT H. sapiens SSL Slorth 0.933062 View
ENSG00000154473 BUB3 ENSG00000157404 KIT H. sapiens SSL Slorth 0.933053 View
ENSG00000093009 CDC45 ENSG00000157404 KIT H. sapiens SSL Slorth 0.933035 View
ENSG00000070831 CDC42 ENSG00000157404 KIT H. sapiens SDL Slorth 0.933026 View
ENSG00000067560 RHOA ENSG00000157404 KIT H. sapiens SSL Slorth 0.93302 View
ENSG00000138829 FBN2 ENSG00000157404 KIT H. sapiens SDL Slorth 0.93299 View
ENSG00000127329 PTPRB ENSG00000157404 KIT H. sapiens SDL Slorth 0.93299 View
ENSG00000134871 COL4A2 ENSG00000157404 KIT H. sapiens SDL Slorth 0.93299 View
ENSG00000063660 GPC1 ENSG00000157404 KIT H. sapiens SDL Slorth 0.932954 View
ENSG00000124164 VAPB ENSG00000157404 KIT H. sapiens SSL Slorth 0.932927 View
ENSG00000115616 SLC9A2 ENSG00000157404 KIT H. sapiens SDL Slorth 0.932121 View
ENSG00000140199 SLC12A6 ENSG00000157404 KIT H. sapiens SDL Slorth 0.932121 View
ENSG00000132155 RAF1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.932114 View