KIT

ENSG00000157404 - H. sapiens

Pathways

Go term Description
GO:0002020 protease binding
GO:0004713 protein tyrosine kinase activity
GO:0004714 transmembrane receptor protein tyrosine kinase activity
GO:0004716 signal transducer, downstream of receptor, with protein tyrosine kinase activity
GO:0005020 stem cell factor receptor activity
GO:0005088 Ras guanyl-nucleotide exchange factor activity
GO:0005515 protein binding
GO:0005524 ATP binding
GO:0019955 cytokine binding
GO:0042803 protein homodimerization activity
GO:0046872 metal ion binding
GO:0046934 phosphatidylinositol-4,5-bisphosphate 3-kinase activity

Drugs

Drug name Description
CABOZANTINIB
DASATINIB Tyrosine-protein kinase ABL inhibitor
IMATINIB Tyrosine-protein kinase ABL inhibitor
LENVATINIB
PAZOPANIB Tyrosine-protein kinase LCK inhibitor
PONATINIB Tyrosine-protein kinase ABL inhibitor
REGORAFENIB Tyrosine-protein kinase ABL inhibitor
SORAFENIB Serine/threonine-protein kinase RAF inhibitor
SUNITINIB Macrophage colony stimulating factor receptor inhibitor

Diseases

Disease Name
GIST
AML
TGCT
mastocytosis
mucosal melanoma
epithelioma

Orthologs

Gene Organism
Pvr D. melanogaster

Related Interactions

Gene ID A Gene Name A Gene ID B Gene Symbol B Organism Source Score?
ENSG00000096063 SRPK1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.871492 View
ENSG00000157404 KIT ENSG00000164924 YWHAZ H. sapiens SSL Slorth 0.871101 View
ENSG00000078043 PIAS2 ENSG00000157404 KIT H. sapiens SSL Slorth 0.87096 View
ENSG00000139842 CUL4A ENSG00000157404 KIT H. sapiens SSL Slorth 0.870709 View
ENSG00000124422 USP22 ENSG00000157404 KIT H. sapiens SSL Slorth 0.870582 View
ENSG00000085733 CTTN ENSG00000157404 KIT H. sapiens SSL Slorth 0.870544 View
ENSG00000102981 PARD6A ENSG00000157404 KIT H. sapiens SSL Slorth 0.870485 View
ENSG00000075785 RAB7A ENSG00000157404 KIT H. sapiens SSL Slorth 0.870158 View
ENSG00000135503 ACVR1B ENSG00000157404 KIT H. sapiens SSL Slorth 0.870152 View
ENSG00000147044 CASK ENSG00000157404 KIT H. sapiens SSL Slorth 0.8687 View
ENSG00000090372 STRN4 ENSG00000157404 KIT H. sapiens SSL Slorth 0.868564 View
ENSG00000119487 MAPKAP1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.86799 View
ENSG00000157404 KIT ENSG00000198742 SMURF1 H. sapiens SSL Slorth 0.867629 View
ENSG00000097007 ABL1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.866983 View
ENSG00000157404 KIT ENSG00000165731 RET H. sapiens SSL Slorth 0.866322 View
ENSG00000047315 POLR2B ENSG00000157404 KIT H. sapiens SSL Slorth 0.866247 View
ENSG00000112685 EXOC2 ENSG00000157404 KIT H. sapiens SSL Slorth 0.866083 View
ENSG00000100347 SAMM50 ENSG00000157404 KIT H. sapiens SSL Slorth 0.865866 View
ENSG00000115085 ZAP70 ENSG00000157404 KIT H. sapiens SSL Slorth 0.865483 View
ENSG00000096717 SIRT1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.863995 View
ENSG00000102882 MAPK3 ENSG00000157404 KIT H. sapiens SSL Slorth 0.863519 View
ENSG00000115808 STRN ENSG00000157404 KIT H. sapiens SSL Slorth 0.863501 View
ENSG00000157404 KIT ENSG00000166501 PRKCB H. sapiens SSL Slorth 0.863283 View
ENSG00000109062 SLC9A3R1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.863047 View
ENSG00000103769 RAB11A ENSG00000157404 KIT H. sapiens SSL Slorth 0.862095 View
ENSG00000065675 PRKCQ ENSG00000157404 KIT H. sapiens SSL Slorth 0.861705 View
ENSG00000136807 CDK9 ENSG00000157404 KIT H. sapiens SSL Slorth 0.861563 View
ENSG00000104695 PPP2CB ENSG00000157404 KIT H. sapiens SSL Slorth 0.861195 View
ENSG00000051180 RAD51 ENSG00000157404 KIT H. sapiens SSL Slorth 0.861141 View
ENSG00000055130 CUL1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.861119 View
ENSG00000129691 ASH2L ENSG00000157404 KIT H. sapiens SSL Slorth 0.860479 View
ENSG00000033327 GAB2 ENSG00000157404 KIT H. sapiens SSL Slorth 0.859009 View
ENSG00000132612 VPS4A ENSG00000157404 KIT H. sapiens SSL Slorth 0.858993 View
ENSG00000134086 VHL ENSG00000157404 KIT H. sapiens SSL Slorth 0.857847 View
ENSG00000143801 PSEN2 ENSG00000157404 KIT H. sapiens SSL Slorth 0.85783 View
ENSG00000071564 TCF3 ENSG00000157404 KIT H. sapiens SSL Slorth 0.857646 View
ENSG00000134602 STK26 ENSG00000157404 KIT H. sapiens SSL Slorth 0.856339 View
ENSG00000064995 TAF11 ENSG00000157404 KIT H. sapiens SSL Slorth 0.856111 View
ENSG00000114867 EIF4G1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.856068 View
ENSG00000140807 NKD1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.855597 View