EP300 - PDGFRA

H. sapiens

SDL interaction

Identifiers

Gene Name Gene ID Diseases Drugs GO terms Orthologs
EP300 ENSG00000100393 colorectal
breast
pancreatic
AML
ALL
DLBCL

No drugs in record

RNA polymerase II core promoter sequence-specific DNA binding
core promoter binding
RNA polymerase II activating transcription factor binding
transcriptional activator activity, RNA polymerase II transcription regulatory region sequence-specific binding
p53 binding
DNA binding
chromatin binding
damaged DNA binding
transcription coactivator activity
histone acetyltransferase activity
lysine N-acetyltransferase activity, acting on acetyl phosphate as donor
protein binding
beta-catenin binding
protein C-terminus binding
transcription factor binding
zinc ion binding
acetyltransferase activity
transferase activity, transferring acyl groups
chromatin DNA binding
activating transcription factor binding
peptide N-acetyltransferase activity
nuclear hormone receptor binding
androgen receptor binding
pre-mRNA intronic binding
BDF1 (S. cerevisiae)
BDF2 (S. cerevisiae)
nej (D. melanogaster)
PDGFRA ENSG00000134853 GIST
idiopathic hypereosinophilic syndrome
paediatric glioblastoma
BECAPLERMIN
LENVATINIB
NINTEDANIB
PAZOPANIB
PONATINIB
REGORAFENIB
SUNITINIB
protein kinase activity
transmembrane receptor protein tyrosine kinase activity
platelet-derived growth factor alpha-receptor activity
vascular endothelial growth factor-activated receptor activity
Ras guanyl-nucleotide exchange factor activity
platelet-derived growth factor receptor binding
protein binding
ATP binding
vascular endothelial growth factor binding
protein homodimerization activity
phosphatidylinositol-4,5-bisphosphate 3-kinase activity
platelet-derived growth factor binding
Pvr (D. melanogaster)